![Improvement of antimalarial activity of a 3-alkylpiridine alkaloid analog by replacing the pyridine ring to a thiazole-containing heterocycle: Mode of action, mutagenicity profile, and Caco-2 cell-based permeability - ScienceDirect Improvement of antimalarial activity of a 3-alkylpiridine alkaloid analog by replacing the pyridine ring to a thiazole-containing heterocycle: Mode of action, mutagenicity profile, and Caco-2 cell-based permeability - ScienceDirect](https://ars.els-cdn.com/content/image/1-s2.0-S0928098719302799-ga1.jpg)
Improvement of antimalarial activity of a 3-alkylpiridine alkaloid analog by replacing the pyridine ring to a thiazole-containing heterocycle: Mode of action, mutagenicity profile, and Caco-2 cell-based permeability - ScienceDirect
Has Ferrocene Really Delivered Its Role in Accentuating the Bioactivity of Organic Scaffolds? | Journal of Medicinal Chemistry
![Antimalarial activity of primaquine operates via a two-step biochemical relay | Nature Communications Antimalarial activity of primaquine operates via a two-step biochemical relay | Nature Communications](https://media.springernature.com/m685/springer-static/image/art%3A10.1038%2Fs41467-019-11239-0/MediaObjects/41467_2019_11239_Fig1_HTML.png)
Antimalarial activity of primaquine operates via a two-step biochemical relay | Nature Communications
![Artemisinin, an Endoperoxide Antimalarial, Disrupts the Hemoglobin Catabolism and Heme Detoxification Systems in Malarial Parasite* - Journal of Biological Chemistry Artemisinin, an Endoperoxide Antimalarial, Disrupts the Hemoglobin Catabolism and Heme Detoxification Systems in Malarial Parasite* - Journal of Biological Chemistry](https://els-jbs-prod-cdn.jbs.elsevierhealth.com/cms/asset/844a8e1c-bff8-4ff4-a045-40461eaa889f/gr1.jpg)
Artemisinin, an Endoperoxide Antimalarial, Disrupts the Hemoglobin Catabolism and Heme Detoxification Systems in Malarial Parasite* - Journal of Biological Chemistry
![Indole based antimalarial compounds targeting the melatonin pathway: Their design, synthesis and biological evaluation - ScienceDirect Indole based antimalarial compounds targeting the melatonin pathway: Their design, synthesis and biological evaluation - ScienceDirect](https://ars.els-cdn.com/content/image/1-s2.0-S0223523419301333-sc1.jpg)
Indole based antimalarial compounds targeting the melatonin pathway: Their design, synthesis and biological evaluation - ScienceDirect
![Antimalarial Inhibitors Targeting Serine Hydroxymethyltransferase (SHMT) with in Vivo Efficacy and Analysis of their Binding Mode Based on X-ray Cocrystal Structures | Journal of Medicinal Chemistry Antimalarial Inhibitors Targeting Serine Hydroxymethyltransferase (SHMT) with in Vivo Efficacy and Analysis of their Binding Mode Based on X-ray Cocrystal Structures | Journal of Medicinal Chemistry](https://pubs.acs.org/cms/10.1021/acs.jmedchem.7b00008/asset/images/large/jm-2017-00008j_0001.jpeg)
Antimalarial Inhibitors Targeting Serine Hydroxymethyltransferase (SHMT) with in Vivo Efficacy and Analysis of their Binding Mode Based on X-ray Cocrystal Structures | Journal of Medicinal Chemistry
![Synthesis, Characterization, and in vitro Antimalarial and Antitumor Activity of New Ruthenium(II) Complexes of Chloroquine | Inorganic Chemistry Synthesis, Characterization, and in vitro Antimalarial and Antitumor Activity of New Ruthenium(II) Complexes of Chloroquine | Inorganic Chemistry](https://pubs.acs.org/cms/10.1021/ic802220w/asset/images/large/ic-2008-02220w_0007.jpeg)
Synthesis, Characterization, and in vitro Antimalarial and Antitumor Activity of New Ruthenium(II) Complexes of Chloroquine | Inorganic Chemistry
![Ikoamide, an Antimalarial Lipopeptide from an Okeania sp. Marine Cyanobacterium | Journal of Natural Products Ikoamide, an Antimalarial Lipopeptide from an Okeania sp. Marine Cyanobacterium | Journal of Natural Products](https://pubs.acs.org/cms/10.1021/acs.jnatprod.9b01147/asset/images/medium/np9b01147_0005.gif)
Ikoamide, an Antimalarial Lipopeptide from an Okeania sp. Marine Cyanobacterium | Journal of Natural Products
![The Antimalarial Natural Product Salinipostin A Identifies Essential α/β Serine Hydrolases Involved in Lipid Metabolism in P. falciparum Parasites - ScienceDirect The Antimalarial Natural Product Salinipostin A Identifies Essential α/β Serine Hydrolases Involved in Lipid Metabolism in P. falciparum Parasites - ScienceDirect](https://ars.els-cdn.com/content/image/1-s2.0-S2451945620300015-fx1.jpg)
The Antimalarial Natural Product Salinipostin A Identifies Essential α/β Serine Hydrolases Involved in Lipid Metabolism in P. falciparum Parasites - ScienceDirect
![Molecular Mechanism of Action of Antimalarial Benzoisothiazolones: Species-Selective Inhibitors of the Plasmodium spp. MEP Pathway enzyme, IspD | Scientific Reports Molecular Mechanism of Action of Antimalarial Benzoisothiazolones: Species-Selective Inhibitors of the Plasmodium spp. MEP Pathway enzyme, IspD | Scientific Reports](https://media.springernature.com/m685/springer-static/image/art%3A10.1038%2Fsrep36777/MediaObjects/41598_2016_Article_BFsrep36777_Fig1_HTML.jpg)
Molecular Mechanism of Action of Antimalarial Benzoisothiazolones: Species-Selective Inhibitors of the Plasmodium spp. MEP Pathway enzyme, IspD | Scientific Reports
![Application of NIR handheld transmission spectroscopy and chemometrics to assess the quality of locally produced antimalarial medicines in the Democratic Republic of Congo - ScienceDirect Application of NIR handheld transmission spectroscopy and chemometrics to assess the quality of locally produced antimalarial medicines in the Democratic Republic of Congo - ScienceDirect](https://ars.els-cdn.com/content/image/1-s2.0-S2666831920300254-fx1.jpg)
Application of NIR handheld transmission spectroscopy and chemometrics to assess the quality of locally produced antimalarial medicines in the Democratic Republic of Congo - ScienceDirect
![Potent Antimalarial 1,2,4‐Trioxanes through Perhydrolysis of Epoxides - Hao - 2013 - Chemistry – A European Journal - Wiley Online Library Potent Antimalarial 1,2,4‐Trioxanes through Perhydrolysis of Epoxides - Hao - 2013 - Chemistry – A European Journal - Wiley Online Library](https://chemistry-europe.onlinelibrary.wiley.com/cms/asset/fe76d1b8-e755-4d88-9d07-ea3d92babb12/mcontent.jpg)
Potent Antimalarial 1,2,4‐Trioxanes through Perhydrolysis of Epoxides - Hao - 2013 - Chemistry – A European Journal - Wiley Online Library
![Antimalarial and anti-inflammatory activities of new chloroquine and primaquine hybrids: Targeting the blockade of malaria parasite transmission - ScienceDirect Antimalarial and anti-inflammatory activities of new chloroquine and primaquine hybrids: Targeting the blockade of malaria parasite transmission - ScienceDirect](https://ars.els-cdn.com/content/image/1-s2.0-S0968089620306623-ga1.jpg)
Antimalarial and anti-inflammatory activities of new chloroquine and primaquine hybrids: Targeting the blockade of malaria parasite transmission - ScienceDirect
Synthesis, Characterization, and in vitro Antimalarial and Antitumor Activity of New Ruthenium(II) Complexes of Chloroquine | Inorganic Chemistry
![Novel Schiff base (E)-2-((4-chloro-3-nitrophenylimino)(phenyl)methyl)-5-methoxyphenol and Mixed Ligand Complexes of Mn(II), Fe(III), Co(II), Ni(II) and Cu(II): synthesis, structure elucidation and potency study as antibacterial, antimalarial ... Novel Schiff base (E)-2-((4-chloro-3-nitrophenylimino)(phenyl)methyl)-5-methoxyphenol and Mixed Ligand Complexes of Mn(II), Fe(III), Co(II), Ni(II) and Cu(II): synthesis, structure elucidation and potency study as antibacterial, antimalarial ...](https://media.springernature.com/lw685/springer-static/image/art%3A10.1007%2Fs13738-021-02431-5/MediaObjects/13738_2021_2431_Figa_HTML.png)
Novel Schiff base (E)-2-((4-chloro-3-nitrophenylimino)(phenyl)methyl)-5-methoxyphenol and Mixed Ligand Complexes of Mn(II), Fe(III), Co(II), Ni(II) and Cu(II): synthesis, structure elucidation and potency study as antibacterial, antimalarial ...
![Preparation and Physicochemical Characterization of an Inclusion Complex Between Dimethylated β-Cyclodextrin and a Drug Lead From a New Class of Orally Active Antimalarial 3,5-Diaryl-2-Aminopyridines - Journal of Pharmaceutical Sciences Preparation and Physicochemical Characterization of an Inclusion Complex Between Dimethylated β-Cyclodextrin and a Drug Lead From a New Class of Orally Active Antimalarial 3,5-Diaryl-2-Aminopyridines - Journal of Pharmaceutical Sciences](https://els-jbs-prod-cdn.jbs.elsevierhealth.com/cms/attachment/be50c221-9b23-4da4-8c72-e7d30cfe0185/gr1_lrg.jpg)
Preparation and Physicochemical Characterization of an Inclusion Complex Between Dimethylated β-Cyclodextrin and a Drug Lead From a New Class of Orally Active Antimalarial 3,5-Diaryl-2-Aminopyridines - Journal of Pharmaceutical Sciences
![Structure-activity and structure-property relationship studies of spirocyclic chromanes with antimalarial activity - ScienceDirect Structure-activity and structure-property relationship studies of spirocyclic chromanes with antimalarial activity - ScienceDirect](https://ars.els-cdn.com/content/image/1-s2.0-S0968089622000219-ga1.jpg)